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Methyltransferase (MTase) Inhibitors
Protein N-terminal MTase 1/2 (NTMT1/2): DC541 (
ACS Med Chem Letts
); GD562; Bisubstrate inhibitors (
PMID: 32605369
); Small molecule inhibitors: GD433 (
PMID:
36634151
)
Nicotinamide N-MTase (NNMT): LL320 (
PMID: 31724854
); II399 (
PMID:
35134268
)
; II559; II630
Protein N-terminal acetyltransferase (NAT) Inhibitors
NatD: YD612 (
PMID:34110812
)
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Our Inhibitors